Pipeline

A Pipeline for
Real Impact.

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Native Complex Platform™ Expanding the Landscape of Druggable GPCRs

At Septerna, we are building a pipeline of highly differentiated GPCR-targeted drug discovery and development programs built on our unique Native Complex Platform™.

We can now reach biologically validated, but historically undruggable GPCRs, as well as the vast majority of unexploited GPCRs still awaiting biological characterization and validation.

The Native Complex Platform™ puts Septerna in a unique position to overcome historical GPCR drug discovery barriers and build a pipeline of new and important medicines for patients.

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Our Pipeline

Target

PTH1R

Mode of Action

Agonist

IND Enabling

Target

TSHR

Mode of Action

Negative Allosteric Modulator

IND Enabling

Target

Target #3

Mode of Action

Agonist

Discovery

Target

Target #4

Mode of Action

Negative Allosteric Modulator

Discovery

Target

New Targets

Mode of Action

Multiple

Discovery

Target

Mode of Action

Discovery

IND Enabling

Clinical

PTH1R

Agonist

TSHR

Negative Allosteric Modulator

Target #3

Agonist

Target #4

Negative Allosteric Modulator

New Targets

Multiple